RANEXA FOR VT
-It might be reasonable to try Ranexa.
-There are small studies that suggest that Ranexa can reduce the
VT burden and ICD shocks in patients with AAD-refracotry VT.
[Bunch, T et al. "Ranolazine reduces ventricular tachycardia
burden and ICD shocks in patients with drug refractory ICD
shocks." Pacing Clin Electrophysiol. 2011 Dec;34(12):1600-6]
-Ranexa could have two main benefits:
(1) It has anti-ischemic effects
(2) It has anti-arrhythmic effects, most likely through
its IKr blockade as well as late INa currents, in
combination with other Class III AADs
-It has been described a possible option for AAD-refractory
ICD shocks secondary to VT
-It is an off-label indication for the drug, and I have
explained this to the patient. He acknowledges this, and is
willing to try it.
-Of note, it is true that Ranexa can potentially prolong the QTc
via blockade of IKr
-Per the MERLIN-TIMI 36 trial, lengthening of the QT
interval has been observed. However, there was no
increased risk of proarrhythmia or SCD observed with
this.
-If Ranexa is started, it might be more reasonable to start with
500 mg po BID given his renal dysfunction